KinasePro

Kinase Chemistry – Just a year and a half behind the times.

ACVR1 + FKBP12

Posted by kinasepro on May 11, 2009

‘nother interesting SGC prerelease

sgc_2

The orange hat on top is FKB12, for which this kind of thing has been seen before w/ TGF-Beta, (1B6C) but this one’s ligated.  I suspect you could infer from this that inhibition of the active site wouldn’t preclude FKBP12 binding…

Leave a comment