Kinase Chemistry – Just a year and a half behind the times.

Archive for January, 2009

Whats that doin there?

Posted by kinasepro on January 20, 2009

Looks like Merck’s released an allosteric CHK1 pdb: 3F9N



Read the rest of this entry »

Posted in Chk1, PDB | 1 Comment »

Plexx in the Black

Posted by kinasepro on January 12, 2009

Possibly unaware of a recent nightclub incident, Roche just put a valuation of 60 million up front for PLX-5568: the ph1 Raf inhibitor.  Likely from the aza-indole genre.

Posted in Plexxikon, RAF | 1 Comment »

Best place to hide a PI3K review?

Posted by kinasepro on January 7, 2009

Somewhere like Biochimica et Biophysica Acta sure would do the trick.

You could also try and bury one somewhere over here or there too…

The BPA one’s good!  Go check it out, thanks VC for the tip.

>> And another one >>  Mol Cancer Ther now in on the act.

Posted in pi3k | 1 Comment »