KinasePro

Kinase Chemistry – Just a year and a half behind the times.

Archive for the ‘Drug Like Properties’ Category

More weekend reading…

Posted by kinasepro on November 4, 2007

Reader RGS really wants you to read AZ’s Nature DD article on Ro5 (mostly clogp/mw)

Astex compiled a table for kinase inhibitors.

GMC has a lot to say on the topic.

KP thinks you can skip today’s lesson if you just stop making 600 mw compounds.

Advertisements

Posted in Drug Like Properties | 5 Comments »

Chemical descriptors of clinical stage kinase inhibitors

Posted by kinasepro on August 25, 2007

– pretty pictures – no data –

Read the rest of this entry »

Posted in Drug Like Properties, General Interest | 2 Comments »

Rule of 5

Posted by kinasepro on August 24, 2007

>> Update: Here.
rule of 5 v 1.0
Read the rest of this entry »

Posted in Drug Like Properties, General Interest | 13 Comments »