KinasePro

Kinase Chemistry – Just a year and a half behind the times.

PF-04217903

Posted by kinasepro on May 12, 2009

This one snuck past me… and into the clinic.  Currently its Ph1 via: WO/2007/132308

OCCN(N=C1)C=C1C2=CN=C(N=NN3CC4=CC=C(N=CC=C5)C5=C4)C3=N2

this and PF-2341066 both still in the pipeline.

note also WO/2007/138472

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One Response to “PF-04217903”

  1. petros said

    It’s also much more selective than PF-2341066

    http://pubs.acs.org/doi/abs/10.1021/bi900438w

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