KinasePro

Kinase Chemistry – Just a year and a half behind the times.

Archive for December 7th, 2007

R-343

Posted by kinasepro on December 7, 2007

Rigel gets 5M & some good news from Pfizer:

Pfizer (NYSE: PFE), has begun a Phase 1 clinical trial of an inhaled formulation of Rigel’s small molecule syk kinase inhibitor, R343, for the treatment of allergic asthma

Posted in Pfizer, Rigel, SYK | 2 Comments »

TG-101348

Posted by kinasepro on December 7, 2007

Targegen’s got a press release:

Plans to initiate a multi-center clinical trial of TG101348, an internally discovered, oral, potent, and highly selective JAK2 inhibitor in January, 2008

A poster at ASH:

…Dual-Acting JAK2/FLT3 Small Molecule Kinase Inhibitor for the Treatment of AML

and some pyrimidines in WO/2007/053452:

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Posted in biotech, clinical, Flt3, JAK | Leave a Comment »