Posted by kinasepro on April 13, 2009
Possibly SAR-502250 its a Mitsubishi / Sanofi TPK1/GSK3 inhibitor:
for Alzheimer’s & Diabetes
This entry was posted on April 13, 2009 at 10:57 pm and is filed under GSK3, Sanofi-Aventis.
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A nice design. No NH is a good thing, for brain penetration.
These days we see quite a few -C-C linkage at 4th position.
This is very unique with morpholin direct substitution at 2nd position. Good rationale of introducing oxadiazole on aryl ring.
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