KinasePro

Kinase Chemistry – Just a year and a half behind the times.

At least its free…

Posted by kinasepro on August 20, 2008

The new ‘Perspective‘: Some useful information bracketed by useless commentary.

Affinity is not even a check-box on the road to an approved drug.  What’s stopping 99.9% of real compounds coming from real programs isn’t potency.  This makes a discussion of how many hydrogen bonds to the hinge are in approved drugs totally irrelevant.

Fact Check:

>> Ruboxistaurin is not an approved drug.

>> Fasudil is only approved in Japan.

>> And you forgot Tasigna

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