Kinase Chemistry – Just a year and a half behind the times.

Archive for July, 2007

PDB Update

Posted by kinasepro on July 3, 2007

2J0K FAK; Harvard, Cell, 129, 1177
2J0M (companion to: 2J0J, 2J0L)

2PTO P38 F169Y Mutant; Locus Discovery; Biochem;
2PV5 P38 D168G mutant (companions to 2pkj, 2ptj)


Posted in PDB | Leave a Comment »


Posted by kinasepro on July 2, 2007

Title’d app is from AstraZeneca and has ’bout 82 thiazoles said to hit c-Fms.


click for the guess Read the rest of this entry »

Posted in Astra, c-fms | 2 Comments »

Chroma Ther. ‘n’ Aurora A

Posted by kinasepro on July 1, 2007

WO/2007/072017 is from ICR and looks a little more polished then the earlier Chroma – quinoline series.


still no candidate though?

Posted in Aurora | Leave a Comment »