KinasePro

Kinase Chemistry – Just a year and a half behind the times.

Pazopanib

Posted by kinasepro on June 19, 2007

aka GW-786034 is GSK’s ‘pan Vegfr’ inhibitor:

O=S(C1=CC(NC2=NC=CC(N(C)C3=CC4=NN(C(C)=C4C=C3)C)=N2)=CC=C1C)(N)=O

salt: hydrochloride
some chemistry here.
clinic: ph iii: RCC, WO/2002/05911

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