Posted by kinasepro on May 17, 2007
Supergen just gave an update in Italy yesterday: webcast here. Skip to ~7 minutes for the kinase portion. The highlight for me is on MP-470 where he says that its uM on met (and ret).
but at AACR last year they suggested that:
In their defence I’ll postulate that they meant 4,000 nM concentrations last year. Ultimately does it matter? Only in so far as how much you can trust what they say… heh