Kinase Chemistry – Just a year and a half behind the times.


Posted by kinasepro on May 2, 2007

Vioquest recently gave an update on their ph i/iia study with this here nucleotide. Nearly as old as ATP itself, the compound was made new again by a diagnostic screen for cancers overexpressing AKT.


Also goes by: API-2, NSC-154020, TCN-P, and triciribine phosphate. and yeh, somebody got the structure wrong in Cancer Res. 04, 4394

(KSR v. Teleflex? suck it.)

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