KinasePro

Kinase Chemistry – Just a year and a half behind the times.

‘Nother “Novel” VEGF candidate

Posted by kinasepro on April 10, 2007

BMS-582664 / Brivanib alaninate

WO/2007/038648 is a development ‘crystalline forms’ application from BMS.

CC(C(OC[C@@H](C)OC([C@@H](C)N)=O)=C1)=C2N1N=CN=C2OC3=C(F)C(C=C(C)N4)=C4C=C3

Discovery: WO/2004/009784. Process: WO/2006/130657. It’s a prodrug / isostere rip on AZD-2171 / Cediranib / Recentin; WO/2000/047212

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