KinasePro

Kinase Chemistry – Just a year and a half behind the times.

Tarceva ®

Posted by kinasepro on April 8, 2007

Tarceva ®, erlotinib hydrochloride, OSI-774

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Discovery: Pfizer WO/1996/30347. Pfizer turned over the rights to OSI to meet U.S. FTC requirements related to Pfizer’s merger with Warner-Lambert in June 2000. The drug is jointly marketted by Genentech, and OSI.
US Approval: November 2004;

PDB: 1M17

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