KinasePro

Kinase Chemistry – Just a year and a half behind the times.

Archive for December 1st, 2006

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Posted by kinasepro on December 1, 2006

Hi Boehringer Ingelhiem, KP likes the BI piperidines/ pyran / cyclohexyl wrinkle on the quinazoline EGF compound series. More derivatives in this continuation, otherwise nothing much to see here.

Move along.

Posted in BI, EGF | Leave a Comment »

US20060270673

Posted by kinasepro on December 1, 2006

Hidy Ho Merck and Co., I’d say nice AKT inhibitors, but I notice you’re doing your xeno studies sub-q.

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Posted in AKT, Merck & Co. | Leave a Comment »

When it rains…

Posted by kinasepro on December 1, 2006

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Posted in Application List | Leave a Comment »

WO2006127961

Posted by kinasepro on December 1, 2006

Hi Scripps, nice indolinones. I don’t generally hit academic patent apps, but for this one… Well for this one – at least someone out there knows why this is a good one to put up.

…Enhanced and unexpected drug like properties that advantageously distinguishes this class of compounds over the known… yada yada yada

alpha-OH > beta-OH

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Posted in SRI, VEGF | 3 Comments »